SCHEMBL13653574

SCHEMBL13653574

CN(C)CCCNc1nc(Nc2ccc(N3CCOCC3)nc2)ncc1C1CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 12/20 0.69
MARK3 P27448 4/20 0.56
IKBKE Q14164 3/20 0.56
CDK2 P24941 2/20 0.56
BRSK2 Q8IWQ3 2/20 0.56
AURKB Q96GD4 2/20 0.56
MKNK1 Q9BUB5 2/20 0.56
IGF1R P08069 1/20 0.50
ULK1 O75385 4/20 0.47
ULK2 Q8IYT8 4/20 0.47
MARK4 Q96L34 2/20 0.46
STK17A Q9UEE5 2/20 0.46
NUAK1 O60285 1/20 0.46
PRKAA2 P54646 1/20 0.46
SIK1 P57059 1/20 0.46
PRKAA1 Q13131 1/20 0.46
MELK Q14680 1/20 0.46
PDK1 Q15118 1/20 0.46
MARK2 Q7KZI7 1/20 0.46
NUAK2 Q9H093 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13460188 0.93 TBK1 (0.67) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3388099 0.89 TBK1 (0.73) TBK1MARK3IKBKECDK2BRSK2
Hydrochloric Acid SCHEMBL3389146 0.89 TBK1 (0.72) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3383970 0.88 TBK1 (0.72) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL13431860 0.87 TBK1 (0.76) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3385005 0.86 TBK1 (0.65) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3388094 0.85 TBK1 (0.75) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3388089 0.85 TBK1 (0.73) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL3383966 0.82 TBK1 (0.71) TBK1MARK3IKBKECDK2BRSK2
SCHEMBL13431843 0.82 TBK1 (1.00) TBK1MARK3IKBKECDK2BRSK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009122180-A1 PYRIMIDINE DERIVATIVES CAPABLE OF INHIBITING ONE OR MORE KINASES MEDICAL RESEARCH COUNCIL (GB) 2009-10-08 WO disclosed