SCHEMBL13655329

SCHEMBL13655329

Nc1ccc2c(c1)-c1sc(C(=O)O)cc1CCO2

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 10/20 0.60
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 3/20 0.52
HPGD P15428 2/20 0.52
GAA P10253 2/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
PIK3CA P42336 8/20 0.50
PIK3CB P42338 4/20 0.50
LMNA P02545 1/20 0.50
GLA P06280 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20597326 0.85 NOTUM (0.77) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL988576 0.85 NOTUM (0.56) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL20597295 0.85 NOTUM (0.77) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL990557 0.83 NOTUM (0.80) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL988949 0.81 PIK3CA (0.63) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL13655403 0.79 PIK3CA (0.70) PIK3CAPIK3CB
SCHEMBL13655350 0.79 NOTUM (0.45) NOTUMKDM4EGAAPIK3CAPIK3CB
SCHEMBL12095162 0.78 NOTUM (0.51) NOTUMKDM4EALDH1A1HPGDGAA
SCHEMBL13655306 0.77 PIK3CA (0.67) PIK3CAPIK3CB
SCHEMBL20596964 0.77 NOTUM (0.70) NOTUMKDM4EALDH1A1GAAPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009123971-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2009-10-08 WO disclosed