SCHEMBL13655350

SCHEMBL13655350

Nc1ccc2c(c1)-c1sc(Br)cc1CCO2

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.45
PIK3CA P42336 13/20 0.39
PIK3CB P42338 4/20 0.39
MAPT P10636 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
DYRK1A Q13627 2/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PRKCI P41743 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12836699 0.89 NOTUM (0.45) NOTUMPIK3CAPIK3CBMAPTKDM4E
SCHEMBL988846 0.81 NOTUM (0.62) NOTUMPIK3CAPIK3CBMAPTKDM4E
SCHEMBL12535860 0.80 PIK3CA (0.52) NOTUMPIK3CAPIK3CB
SCHEMBL13655329 0.79 NOTUM (0.60) NOTUMPIK3CAPIK3CBKDM4EGAA
SCHEMBL988650 0.76 PIK3CA (0.43) NOTUMPIK3CAPIK3CB
SCHEMBL1484768 0.71 PIK3CA (0.52) NOTUMPIK3CAPIK3CB
SCHEMBL379230 0.70 PRKCI (0.56) MAPTKDM4EGAADYRK1ARAB9A
SCHEMBL29364809 0.70 PRKCI (0.56) MAPTKDM4EGAADYRK1ARAB9A
SCHEMBL988463 0.70 NOTUM (0.70) NOTUMPIK3CAPIK3CBKDM4EGAA
SCHEMBL1484735 0.69 MAP3K14 (0.40) NOTUMPIK3CAPIK3CBMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009123971-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2009-10-08 WO disclosed