SCHEMBL13655398

SCHEMBL13655398

Nc1ccc2c(c1)OCCc1cc(-c3n[nH]cc3-c3ccccc3Cl)sc1-2

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 19/20 0.59
PIK3CB P42338 5/20 0.40
NOTUM Q6P988 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1040905 0.90 PIK3CA (0.65) PIK3CAPIK3CBNOTUM
SCHEMBL1038149 0.89 PIK3CA (0.54) PIK3CAPIK3CBNOTUM
SCHEMBL1040682 0.87 PIK3CA (0.70) PIK3CAPIK3CBNOTUM
SCHEMBL1041570 0.86 PIK3CA (0.52) PIK3CAPIK3CBNOTUM
SCHEMBL12535914 0.85 PIK3CA (0.61) PIK3CAPIK3CB
SCHEMBL990580 0.74 PIK3CA (1.00) PIK3CAPIK3CBNOTUM
SCHEMBL13655399 0.74 PIK3CA (0.82) PIK3CAPIK3CB
SCHEMBL1039507 0.74 PIK3CA (0.71) PIK3CAPIK3CB
SCHEMBL990834 0.74 PIK3CA (0.70) PIK3CAPIK3CBNOTUM
SCHEMBL991296 0.74 PIK3CA (0.82) PIK3CAPIK3CBNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009123971-A1 BENZOPYRAN AND BENZOXEPIN PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH, INC. (US) 2009-10-08 WO disclosed