SCHEMBL13655584

SCHEMBL13655584

CO[C@@]1(C)CC(C)C(=O)C(C)[C@H]2N(CCCCn3cnc(-c4cccnc4)c3)C(=O)OC23C(OC(=O)C(C)C(=O)C(C)[C@H]1OC(=O)C1CN(C(=O)OC(C)(C)C)C(C)(C)O1)[C@@H]3C

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
ABCC4 O15439 1/20 0.53
ABCB11 O95342 1/20 0.53
CYP3A5 P20815 1/20 0.53
PTGS1 P23219 1/20 0.53
CYP3A7 P24462 1/20 0.53
KCNH2 Q12809 1/20 0.53
CYP3A43 Q9HB55 1/20 0.53
SLCO1B3 Q9NPD5 1/20 0.53
SLCO1B1 Q9Y6L6 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL784958 0.91 CYP3A4 (0.64) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL799508 0.83 CYP3A4 (0.61) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL13655585 0.83 CYP3A4 (0.61) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL13655659 0.83 CYP3A4 (0.59) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL13655658 0.83 CYP3A4 (0.48) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL799164 0.81 CYP3A4 (0.58) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL10270380 0.75 CYP3A4 (0.65) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL12254525 0.74 CYP3A4 (0.72) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL9968998 0.73 CYP3A4 (0.73) CYP3A4ABCC4ABCB11CYP3A5PTGS1
SCHEMBL784787 0.73 CYP3A4 (0.76) CYP3A4ABCC4ABCB11CYP3A5PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601695-B2 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal OPTIMER PHARMACEUTICALS, INC. (US) 2009-10-13 US disclosed