SCHEMBL13655603

SCHEMBL13655603

Cc1cc(I)c(I)c(C(=O)OCCC(C)(C)C(C)(C)C)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.35
TSHR P16473 4/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPK1 P28482 1/20 0.32
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
ALDH1A1 P00352 3/20 0.31
KMT2A Q03164 2/20 0.31
LMNA P02545 1/20 0.31
EGFR P00533 1/20 0.31
MEN1 O00255 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13655561 0.87 HDAC3 (0.39) ESR1TSHRTDP1L3MBTL1ALDH1A1
SCHEMBL22014584 0.82 ESR1 (0.35) ESR1TSHRTDP1L3MBTL1TP53
SCHEMBL21730572 0.79 TSHR (0.48) TSHRL3MBTL1CYP3A4MAPK1ALDH1A1
SCHEMBL21842558 0.75 TSHR (0.41) ESR1TSHRTDP1L3MBTL1TP53
SCHEMBL13655604 0.71 HDAC3 (0.37) KMT2ALMNAMEN1HDAC3HDAC4
SCHEMBL26229419 0.70 MEN1 (0.33) KMT2AMEN1
SCHEMBL22006102 0.69 CNR2 (0.30) CNR2
SCHEMBL26426586 0.67 HDAC3 (0.36) ESR1TSHRCYP3A4ALDH1A1KMT2A
SCHEMBL22640242 0.67 HDAC3 (0.36) ESR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL26343120 0.67 HDAC3 (0.36) ESR1HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090252678-A1 COX-2-TARGETED IMAGING AGENTS VANDERBILT UNIVERSITY (US) 2009-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090252678-A1 COX-2-TARGETED IMAGING AGENTS PTGS2, PTGES2, PTGER2 ESR1 1247/4885TSHR 3905/4885TDP1 3827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.