SCHEMBL13655749

SCHEMBL13655749

CN(C(=O)N1CC(c2cc(F)ccc2F)=CC1c1cccc(O)c1)C1CCOC1

nearest known ligand 0.76

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 19/20 0.76
KCNH2 Q12809 14/20 0.76

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4062461 1.00 KIF11 (0.76) KIF11KCNH2
SCHEMBL4060646 0.95 KIF11 (0.80) KIF11KCNH2
SCHEMBL13655793 0.95 KIF11 (0.80) KIF11KCNH2
SCHEMBL4057419 0.92 KIF11 (0.75) KIF11KCNH2
SCHEMBL4060410 0.86 KIF11 (1.00) KIF11KCNH2
SCHEMBL14277511 0.86 KIF11 (0.57) KIF11KCNH2
SCHEMBL5104349 0.86 KIF11 (0.57) KIF11KCNH2
SCHEMBL4057497 0.86 KIF11 (1.00) KIF11KCNH2
SCHEMBL4063819 0.86 KIF11 (1.00) KIF11KCNH2
SCHEMBL4059744 0.85 KIF11 (0.72) KIF11KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1515724-B1 MITOTIC KINESIN INHIBITORS MERCK & CO INC (US) 2009-10-21 EP disclosed
US-7348440-B2 Kinesin spindle protein (KSP) inhibitors, e.g., 4-(2,5-Difluorophenyl)-N-[(3S,4S)-3-fluoropiperidin-4-yl]-2-hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1N-pyrrole-1-carboxamide, and a carrier; antiproliferative and -carcinogenic agents; side effects reduction; used with an estrogen receptor modulator MERCK & CO., INC. (US) 2008-03-25 US disclosed