SCHEMBL1365690

SCHEMBL1365690

O=C(CS)NCCCCCNC(=O)c1cnc2ccccc2c1

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 14/20 0.67
HDAC10 Q969S8 12/20 0.67
HDAC6 Q9UBN7 12/20 0.67
HDAC2 Q92769 12/20 0.67
HDAC3 O15379 11/20 0.67
HDAC8 Q9BY41 11/20 0.67
HDAC4 P56524 9/20 0.67
HDAC7 Q8WUI4 9/20 0.67
HDAC11 Q96DB2 9/20 0.67
HDAC9 Q9UKV0 9/20 0.67
HDAC5 Q9UQL6 9/20 0.67
DRD2 P14416 3/20 0.54
DRD3 P35462 3/20 0.54
HTR1A P08908 1/20 0.54
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
TNKS O95271 1/20 0.50
PPARD Q03181 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2639346 0.84 MGAM (0.56) HDAC1HDAC10HDAC6HDAC2HDAC3
SCHEMBL5020897 0.84 HDAC3 (0.61) HDAC1HDAC2HDAC3DRD2DRD3
SCHEMBL10242977 0.82 HDAC3 (0.61) HDAC1HDAC2HDAC3DRD2DRD3
SCHEMBL29222038 0.79 HDAC3 (0.61) HDAC1HDAC2HDAC3DRD2DRD3
SCHEMBL30858823 0.79 HDAC3 (0.61) HDAC1HDAC2HDAC3DRD2DRD3
SCHEMBL2639342 0.79 PPARD (0.57) HDAC1HDAC2HDAC3DRD2DRD3
SCHEMBL1937005 0.78 HDAC1 (1.00) HDAC1HDAC2HDAC3
SCHEMBL28408662 0.77 HDAC6 (0.74) HDAC1HDAC10HDAC6HDAC2HDAC3
SCHEMBL10207276 0.77 HDAC1 (1.00) HDAC1HDAC10HDAC6HDAC2HDAC3
SCHEMBL1364346 0.77 HDAC1 (0.76) HDAC1HDAC10HDAC6HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8067600-B2 Histone deacetylase inhibitors and methods of use thereof GEORGETOWN UNIVERSITY (US) 2011-11-29 US disclosed
US-8067600-B2 Histone deacetylase inhibitors and methods of use thereof GEORGETOWN UNIVERSITY (US) 2011-11-29 US disclosed
US-8067600-B2 Histone deacetylase inhibitors and methods of use thereof GEORGETOWN UNIVERSITY (US) 2011-11-29 US disclosed
US-7507828-B2 Histone deacetylase inhibitors and methods of use thereof GEORGETOWN UNIVERSITY (US) 2009-03-24 US disclosed
US-7507828-B2 Histone deacetylase inhibitors and methods of use thereof GEORGETOWN UNIVERSITY (US) 2009-03-24 US disclosed