SCHEMBL1365778

SCHEMBL1365778

CCC(c1ncc[nH]1)n1c(C)c(C(=O)N[C@H](c2cccc(F)c2)C2CCC2)c2cccc(F)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.42
TACR3 P29371 10/20 0.39
PDE2A O00408 3/20 0.33
SMYD3 Q9H7B4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1364771 0.97 CYP2C9 (0.45) CYP2C9TACR3PDE2A
SCHEMBL1365500 0.91 CYP2C9 (0.43) CYP2C9TACR3PDE2A
SCHEMBL2357653 0.86 CYP2C9 (0.34) CYP2C9TACR3
SCHEMBL1366497 0.84 CYP2C9 (0.43) CYP2C9TACR3PDE2A
SCHEMBL1364412 0.81 CYP2C9 (0.45) CYP2C9TACR3PDE2A
SCHEMBL1364883 0.81 CYP2C9 (0.45) CYP2C9TACR3PDE2A
SCHEMBL1364900 0.81 CYP2C9 (0.46) CYP2C9TACR3PDE2A
SCHEMBL7949895 0.80 CYP2C9 (0.52) CYP2C9TACR3PDE2A
SCHEMBL7942563 0.79 CYP2C9 (0.47) CYP2C9TACR3PDE2ASMYD3
SCHEMBL16566393 0.79 CYP2C9 (0.47) CYP2C9TACR3PDE2ASMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-11-24 US claimed
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2011-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110288120-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS KCNK3, KCNQ3, KCNN3 CYP2C9 2420/4885TACR3 36/4885PDE2A 691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.