SCHEMBL13658302

SCHEMBL13658302

CNc1cc(C)ncc1N

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
UHRF1 Q96T88 1/20 0.56
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
PRKCI P41743 1/20 0.32
AOC1 P19801 1/20 0.32
AOC3 Q16853 1/20 0.32
NOS3 P29474 3/20 0.32
NOS2 P35228 3/20 0.32
NOS1 P29475 2/20 0.32
NNMT P40261 1/20 0.31
MAP4K4 O95819 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18624692 0.83 UHRF1 (0.50) UHRF1CYP1A2CYP2A6PRKCIAOC1
SCHEMBL11581586 0.80 HDAC1 (0.37) UHRF1PRKCIAOC1AOC3MAP4K4
SCHEMBL12706566 0.77 UHRF1 (0.43) UHRF1CYP1A2CYP2A6AOC1AOC3
SCHEMBL30711414 0.77 UHRF1 (0.39) UHRF1PRKCIAOC1AOC3MAP4K4
SCHEMBL10233595 0.77 UHRF1 (0.34) UHRF1PRKCIAOC1AOC3MAP4K4
SCHEMBL10110103 0.77 UHRF1 (0.34) UHRF1PRKCIAOC1AOC3MAP4K4
SCHEMBL1584807 0.77 UHRF1 (0.39) UHRF1PRKCIAOC1AOC3MAP4K4
SCHEMBL12456743 0.77 UHRF1 (0.34) UHRF1PRKCIAOC1AOC3NNMT
Hydrochloric Acid SCHEMBL20266526 0.75 UHRF1 (0.38) UHRF1PRKCIAOC1AOC3EGFR
SCHEMBL23181522 0.74 UHRF1 (0.35) UHRF1CYP1A2CYP2A6NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2313412-B1 NOVEL DERIVATIVES OF PYRROLOINDOLE INHIBITORS OF HSP90, COMPOSITIONS CONTAINING SAME, AND USE THEREOF SANOFI SA (FR) 2013-01-02 EP disclosed
WO-2009122034-A2 NOVEL HSP90 INHIBITORY CARBAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME, AND USE THEREOF SANOFI-AVENTIS (FR) 2009-10-08 WO disclosed