SCHEMBL23181522

SCHEMBL23181522

CNc1cc(C)ncc1F

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
UHRF1 Q96T88 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34
NPC1 O15118 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
SLC6A4 P31645 1/20 0.33
RPS6KA3 P51812 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
RAB9A P51151 1/20 0.32
DAO P14920 1/20 0.32
LYN P07948 2/20 0.31
BTK Q06187 2/20 0.31
FEN1 P39748 1/20 0.30
NOS3 P29474 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12706566 0.77 UHRF1 (0.43) UHRF1CYP1A2CYP2A6SLC6A4NOS3
SCHEMBL19462480 0.77 TGFBR1 (0.38) KCNQ3KCNQ2DAO
SCHEMBL28897534 0.77 CTSD (0.31)
SCHEMBL5514290 0.75 HSD17B10 (0.34) LYNBTK
SCHEMBL13658302 0.74 UHRF1 (0.56) UHRF1CYP1A2CYP2A6NOS3NOS2
SCHEMBL20931323 0.74 SLC6A2 (0.36) UHRF1CYP1A2CYP2A6SLC6A4DAO
SCHEMBL25669006 0.74
SCHEMBL31099115 0.74 MAPK8 (0.39) RPS6KA3
SCHEMBL1746425 0.73 UHRF1 (0.48) UHRF1CYP1A2CYP2A6SLC6A4NOS3
SCHEMBL18010004 0.72 PSIP1 (0.49) FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023064585-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed
WO-2023064584-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY (US) 2023-04-20 WO disclosed
WO-2021057975-A1 MUTANT IDH2 INHIBITOR AND APPLICATION THEREOF 贝达药业股份有限公司 2021-04-01 WO disclosed