SCHEMBL13658397

SCHEMBL13658397

Cc1cc(-n2c3ccccc3c3c(-c4nc5ccc(F)cc5[nH]4)cccc32)cnc1C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 3/20 0.39
CHEK2 O96017 8/20 0.39
SYK P43405 1/20 0.38
LRRK2 Q5S007 1/20 0.38
TSSK3 Q96PN8 1/20 0.38
F7 P08709 1/20 0.37
METAP2 P50579 1/20 0.37
METAP1 P53582 1/20 0.37
CBFB Q13951 1/20 0.37
F2 P00734 1/20 0.36
F10 P00742 1/20 0.36
PLG P00747 1/20 0.36
PLAU P00749 1/20 0.36
PLAT P00750 1/20 0.36
PRSS1 P07477 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2184585 0.85 HSP90AA1 (0.44) CHEK2SYKLRRK2TSSK3
SCHEMBL12411763 0.84 JAK2 (0.41) CHEK2SYKLRRK2TSSK3
SCHEMBL12411776 0.84 CHEK2 (0.37) AMY1ACHEK2SYKLRRK2TSSK3
SCHEMBL2185941 0.82 CHEK2 (0.42) AMY1ACHEK2F7F2F10
SCHEMBL2182351 0.81 CHEK2 (0.46) CHEK2F7F2F10PLG
SCHEMBL2182007 0.81 CHEK2 (0.41) AMY1ACHEK2F7METAP2METAP1
SCHEMBL13658326 0.78 HSP90AA1 (0.48)
SCHEMBL2180286 0.78 AMY1A (0.40) AMY1ACHEK2F2F10PLG
SCHEMBL2180934 0.77 CHEK2 (0.37) AMY1ACHEK2F7HDAC6
SCHEMBL2181385 0.77 HSP90AA1 (0.42) AMY1ACHEK2F7KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009122034-A2 NOVEL HSP90 INHIBITORY CARBAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME, AND USE THEREOF SANOFI-AVENTIS (FR) 2009-10-08 WO disclosed