SCHEMBL13660310

SCHEMBL13660310

O=c1c2ncccc2nc([C@@H]2C[C@@H]3C[C@@H]3C2)n1-c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.42
PDE4B Q07343 1/20 0.40
PDE4D Q08499 1/20 0.40
SCN9A Q15858 3/20 0.38
TSHR P16473 1/20 0.36
EP300 Q09472 1/20 0.36
CREBBP Q92793 1/20 0.36
KAT2A Q92830 1/20 0.36
KAT2B Q92831 1/20 0.36
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
RECQL P46063 1/20 0.35
TOP1 P11387 2/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD11B1 P28845 1/20 0.35
POLB P06746 1/20 0.34
FABP1 P07148 1/20 0.34
AOC3 Q16853 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13660416 0.88 HRH3 (0.42) HRH3PDE4BPDE4DTSHREP300
SCHEMBL3169447 0.82 SCN9A (0.40) HRH3PDE4BPDE4DSCN9AEP300
SCHEMBL3169440 0.82 SCN9A (0.40) HRH3PDE4BPDE4DSCN9AEP300
SCHEMBL13660311 0.82 HRH3 (0.40) HRH3PDE4BPDE4DSCN9AEP300
SCHEMBL13660459 0.81 PDE4B (0.46) HRH3PDE4BPDE4DTSHRPIK3CD
SCHEMBL13660456 0.78 HRH3 (0.40) HRH3PDE4BPDE4DTSHREP300
SCHEMBL13660412 0.78 HRH3 (0.40) HRH3PDE4BPDE4DTSHREP300
SCHEMBL11920282 0.76 EP300 (0.41) HRH3PDE4BPDE4DTSHREP300
SCHEMBL2233132 0.76 PDE4B (0.43) HRH3PDE4BPDE4DTSHREP300
SCHEMBL13660461 0.74 HRH3 (0.37) HRH3PDE4BPDE4DPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO disclosed