SCHEMBL13660459

SCHEMBL13660459

N#Cc1ccc(-n2c([C@@H]3C[C@@H]4C[C@@H]4C3)nc3cccnc3c2=O)cn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 5/20 0.46
PDE4D Q08499 3/20 0.46
USP14 P54578 2/20 0.41
HRH3 Q9Y5N1 1/20 0.39
PDE4A P27815 2/20 0.37
SLC40A1 Q9NP59 2/20 0.34
PIK3CD O00329 5/20 0.33
PDE4C Q08493 1/20 0.32
PIK3CG P48736 3/20 0.32
PIK3CA P42336 1/20 0.32
PDE10A Q9Y233 2/20 0.32
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
PIK3CB P42338 1/20 0.30
TSHR P16473 1/20 0.30
GFER P55789 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13660309 0.88 PDE4B (0.43) PDE4BPDE4DUSP14HRH3PDE4A
SCHEMBL13660312 0.88 PDE4B (0.43) PDE4BPDE4DUSP14HRH3PDE4A
SCHEMBL13660313 0.84 PDE4B (0.44) PDE4BPDE4DUSP14HRH3PDE4A
SCHEMBL3169708 0.84 PDE4B (0.44) PDE4BPDE4DUSP14HRH3PDE4A
SCHEMBL3169713 0.84 PDE4B (0.44) PDE4BPDE4DUSP14HRH3PDE4A
SCHEMBL13660310 0.81 HRH3 (0.42) PDE4BPDE4DHRH3PIK3CDTSHR
SCHEMBL13660416 0.81 HRH3 (0.42) PDE4BPDE4DUSP14HRH3PIK3CD
SCHEMBL13660461 0.73 HRH3 (0.37) PDE4BPDE4DUSP14HRH3
SCHEMBL13660463 0.73 PDE4B (0.37) PDE4BPDE4DUSP14HRH3
SCHEMBL3174425 0.70 PDE4B (0.36) PDE4BPDE4DUSP14HRH3PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009121036-A2 SUBSTITUTED ARYL PYRIMIDINONE DERIVATIVES NEUROGEN CORPORATION (US) 2009-10-01 WO disclosed