SCHEMBL13664

SCHEMBL13664

Cc1cccnc1-c1ccc2nc3c(cc2c1)CC(C(=O)NCCC(C)(C)C)N3

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 8/20 0.57
CTSD P07339 2/20 0.57
ABL1 P00519 2/20 0.41
GRIA2 P42262 1/20 0.38
PDK1 Q15118 5/20 0.35
PDK2 Q15119 5/20 0.35
PDK3 Q15120 5/20 0.35
PDK4 Q16654 5/20 0.35
SSTR4 P31391 3/20 0.34
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13645 0.77 BACE1 (0.33) BACE1CTSD
SCHEMBL9166 0.72 BACE1 (1.00) BACE1CTSD
SCHEMBL9061 0.72 BACE1 (1.00) BACE1CTSD
SCHEMBL14321300 0.66 BACE1 (0.65) BACE1CTSDABL1TRPV1
SCHEMBL9702 0.66 BACE1 (0.87) BACE1CTSD
SCHEMBL14321873 0.65 BACE1 (0.69) BACE1CTSD
SCHEMBL17620320 0.64 BACE1 (0.79) BACE1CTSD
SCHEMBL9396 0.64 BACE1 (0.48) BACE1CTSD
SCHEMBL8994 0.63 BACE1 (1.00) BACE1CTSD
SCHEMBL14321762 0.63 BACE1 (1.00) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063233-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed