SCHEMBL13645

SCHEMBL13645

CC1CC1c1ccc2nc3c(cc2c1)CC(C(=O)NCCC(C)(C)C)N3

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 6/20 0.33
TLR9 Q9NR96 1/20 0.32
TLR8 Q9NR97 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
CTSD P07339 2/20 0.31
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13664 0.77 BACE1 (0.57) BACE1CTSD
SCHEMBL9125 0.72 BACE1 (0.62) BACE1CTSD
SCHEMBL17620302 0.72 BACE1 (0.62) BACE1CTSD
SCHEMBL14324954 0.63 ALDH1A1 (0.36)
SCHEMBL14324953 0.63 ALDH1A1 (0.36)
SCHEMBL17620319 0.62 BACE1 (0.59) BACE1CTSD
SCHEMBL15541599 0.56 SIGMAR1 (0.38) SIGMAR1
SCHEMBL18555901 0.55 CTSC (0.43) SIGMAR1
SCHEMBL16464588 0.54 CHIA (0.39)
SCHEMBL16464589 0.54 CHIA (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063233-A1 AMINO HETEROARYL COMPOUNDS AS BETA-SECRETASE MODULATORS AND METHODS OF USE AMGEN INC. (US) 2011-05-26 WO disclosed