SCHEMBL13664886

SCHEMBL13664886

C=N/C(=C\C=C/C)c1cc(N)ccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.35
TSHR P16473 1/20 0.35
P2RX7 Q99572 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25166279 0.80 P2RX7 (0.38) CYP3A4P2RX7
SCHEMBL24785949 0.73
SCHEMBL19651204 0.67 P2RX7 (0.40) CYP3A4TSHRP2RX7
SCHEMBL13689798 0.67 CYP3A4 (0.48) CYP3A4TSHRP2RX7CA1CA2
SCHEMBL17263342 0.64 CYP3A4 (0.50) CYP3A4TSHRP2RX7CA1CA2
SCHEMBL20076361 0.64 CYP3A4 (0.50) CYP3A4TSHRP2RX7CA1CA2
SCHEMBL21021855 0.64 CYP3A4 (0.32) CYP3A4TSHRP2RX7
SCHEMBL19101609 0.64 TSHR (0.32) CYP3A4TSHR
SCHEMBL1099858 0.63 CYP3A4 (0.48) CYP3A4TSHRP2RX7CA1CA2
SCHEMBL2553178 0.63 CYP3A4 (0.48) CYP3A4TSHRP2RX7CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009126863-A2 PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING GENENTECH, INC. (US) 2009-10-15 WO disclosed