SCHEMBL13667331

SCHEMBL13667331

CC(C)(C)OC(=O)N[C@@H](CCOc1cccc(Br)c1)C(=O)OC1CCCC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 5/20 0.52
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
AAK1 Q2M2I8 2/20 0.42
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 3/20 0.41
RAB9A P51151 1/20 0.40
LNPEP Q9UIQ6 1/20 0.39
KLK7 P49862 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL193352 0.89 CACNA1B (0.52) CACNA1BAAK1KDM4EALDH1A1KLK7
SCHEMBL193351 0.89 CACNA1B (0.52) CACNA1BAAK1KDM4EALDH1A1KLK7
SCHEMBL10052884 0.88 CACNA1B (0.60) CACNA1BCTSSCTSKAAK1ALDH1A1
SCHEMBL193656 0.85 CACNA1B (0.49) CACNA1BRAB9AMEN1KMT2APOLB
SCHEMBL193655 0.85 CACNA1B (0.49) CACNA1BRAB9AMEN1KMT2APOLB
SCHEMBL1147671 0.84 CACNA1B (0.47) CACNA1BAAK1KLK7
SCHEMBL490684 0.83 CACNA1B (0.59) CACNA1BCTSSCTSKAAK1ALDH1A1
SCHEMBL192979 0.83 CACNA1B (0.54) CACNA1BALDH1A1KLK7LMNA
SCHEMBL192978 0.83 CACNA1B (0.54) CACNA1BALDH1A1KLK7LMNA
SCHEMBL8257659 0.82 CACNA1B (0.51) CACNA1BAAK1KLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130434-A1 INHIBITORS OF IKK-β SERINE-THREONINE PROTEIN KINASE CHROMA THERAPEUTICS LTD. (GB) 2009-10-29 WO disclosed