SCHEMBL13670443

SCHEMBL13670443

CC1CCc2nc(S)c(C#N)cc2C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.38
ALDH1A1 P00352 10/20 0.38
GLA P06280 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 4/20 0.36
LMNA P02545 2/20 0.36
HSD17B10 Q99714 3/20 0.36
HTT P42858 3/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4705570 0.82 MAPT (0.37) KDM4EALDH1A1SMN1; SMN2HSD17B10HTT
SCHEMBL4701697 0.82 KDM4E (0.40) KDM4EALDH1A1SMN1; SMN2HSD17B10HTT
SCHEMBL7999907 0.80 KDM4E (0.63) KDM4EALDH1A1SMN1; SMN2TP53LMNA
SCHEMBL5242785 0.78 ALDH1A1 (0.36) KDM4EALDH1A1GLASMN1; SMN2HSD17B10
SCHEMBL4703102 0.74 KDM4E (0.35) KDM4EALDH1A1SMN1; SMN2HSD17B10MEN1
SCHEMBL4705550 0.73 KDM4E (0.42) KDM4ESMN1; SMN2GAAPOLB
SCHEMBL14955079 0.73 SMN1; SMN2 (0.63) KDM4EALDH1A1SMN1; SMN2HSD17B10HTT
SCHEMBL14954856 0.72 MAPT (0.50) KDM4EALDH1A1SMN1; SMN2TP53LMNA
SCHEMBL29741226 0.71 SMN1; SMN2 (0.59) KDM4EALDH1A1GLASMN1; SMN2TP53
SCHEMBL4705401 0.69 POLB (0.37) KDM4EALDH1A1SMN1; SMN2HSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608643-B2 Compounds for inhibiting KSP kinesin activity SCHERING CORPORATION (US) 2009-10-27 US disclosed