SCHEMBL13675004

SCHEMBL13675004

Nc1cc(CF)cc(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.45
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
MAOB P27338 4/20 0.38
TAAR1 Q96RJ0 1/20 0.37
NR2E1 Q9Y466 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
KIF11 P52732 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
TACR1 P25103 3/20 0.33
PTPN5 P54829 1/20 0.33
CACNA1F O60840 1/20 0.33
CACNA1D Q01668 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL864911 0.84 IDO1 (0.47) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL5776968 0.84 IDO1 (0.54) IDO1TSHRTAAR1TACR1CACNA1F
SCHEMBL2793814 0.83 TAAR1 (0.43) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL10200704 0.83 IDO1 (0.45) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL10959537 0.81 IDO1 (0.44) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL29467109 0.81 IDO1 (0.44) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL129085 0.81 RXRA (0.45) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL2793246 0.80 TAAR1 (0.41) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL2795945 0.80 TAAR1 (0.41) IDO1TSHRMAPK1MAOBTAAR1
SCHEMBL806196 0.79 TAAR1 (0.56) IDO1TSHRMAPK1MAOBTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601725-B2 Thienopyrimidines useful as Aurora kinase inhibitors SUNESIS PHARMACEUTICALS, INC. (US) 2009-10-13 US disclosed