SCHEMBL13675170

SCHEMBL13675170

Cc1cccc(Nc2ncnc3nc(Nc4ccccc4)sc23)c1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.74
HTT P42858 3/20 0.52
MAPK1 P28482 2/20 0.52
TSHR P16473 1/20 0.52
RAB9A P51151 1/20 0.52
GFER P55789 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HIF1A Q16665 1/20 0.51
TRPV1 Q8NER1 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49
CHRNA7 P36544 1/20 0.47
CDK1 P06493 1/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13672688 0.86 EGFR (1.00) EGFRCDK1
SCHEMBL13675197 0.86 EGFR (0.75) EGFRTRPV1CHRNA7
SCHEMBL13672701 0.85 EGFR (1.00) EGFRTRPV1CDK1
SCHEMBL13672700 0.85 EGFR (0.74) EGFRTRPV1
SCHEMBL13674977 0.85 EGFR (0.65) EGFRHTTMAPK1TSHRRAB9A
SCHEMBL13672705 0.81 EGFR (0.84) EGFRTRPV1CDK1
SCHEMBL13675243 0.80 EGFR (0.77) EGFR
SCHEMBL13674985 0.79 EGFR (0.75) EGFRTRPV1CHRNA7
SCHEMBL13672699 0.79 EGFR (1.00) EGFRTRPV1CDK1
SCHEMBL5134221 0.76 EGFR (1.00) EGFRHTTRAB9ATRPV1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7605154-B2 ATP-protein kinase inhibitors; cytomegalovirus; contraceptive agents; cancer; N7-(3-ethynyl-phenyl)-N2-(4-piperidin-1-ylmethyl-phenyl)-thiazolo[4,5-d]pyrimidine-2,7-diamine JANSSEN PHARMACEUTICA N.V. (BE) 2009-10-20 US disclosed