SCHEMBL13675197

SCHEMBL13675197

Cc1cc(Cl)cc(Nc2ncnc3nc(Nc4ccccc4)sc23)c1

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 0.75
TRPV1 Q8NER1 2/20 0.49
CHRNA7 P36544 1/20 0.45
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13672705 0.92 EGFR (0.84) EGFRTRPV1ADORA3ADORA2A
SCHEMBL13672701 0.86 EGFR (1.00) EGFRTRPV1
SCHEMBL13675170 0.86 EGFR (0.74) EGFRTRPV1CHRNA7
SCHEMBL13675044 0.84 EGFR (0.75) EGFRTRPV1
SCHEMBL14462166 0.84 EGFR (0.71) EGFRTRPV1ADORA3ADORA2A
SCHEMBL13672699 0.80 EGFR (1.00) EGFRTRPV1
SCHEMBL13672700 0.76 EGFR (0.74) EGFRTRPV1ADORA3ADORA2A
SCHEMBL5066710 0.76 EGFR (0.83) EGFRTRPV1
SCHEMBL13675051 0.75 EGFR (0.78) EGFRTRPV1
SCHEMBL4479462 0.75 EGFR (0.64) EGFRTRPV1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7605154-B2 ATP-protein kinase inhibitors; cytomegalovirus; contraceptive agents; cancer; N7-(3-ethynyl-phenyl)-N2-(4-piperidin-1-ylmethyl-phenyl)-thiazolo[4,5-d]pyrimidine-2,7-diamine JANSSEN PHARMACEUTICA N.V. (BE) 2009-10-20 US disclosed