SCHEMBL13675226

SCHEMBL13675226

C=CCN(CC(=O)OC)S(=O)(=O)c1sc(C(CC)(CC)c2ccc(O)c(C)c2)cc1C

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 16/20 0.38
ESR2 Q92731 5/20 0.38
AR P10275 3/20 0.38
VDR P11473 1/20 0.35
HDAC3 O15379 2/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13672897 0.86 HDAC3 (0.36) VDRHDAC3HDAC6
SCHEMBL13366780 0.85 VDR (0.50) ARVDRHDAC3
SCHEMBL13675225 0.76 ESR1 (0.45) ESR1ESR2ARVDR
SCHEMBL3392747 0.73 ESR1 (0.44) ESR1ESR2ARVDRHDAC3
SCHEMBL13675224 0.72 ESR1 (0.54) ESR1ESR2ARVDR
SCHEMBL3391928 0.70 ESR1 (0.46) ESR1ESR2ARVDR
SCHEMBL13366679 0.70 ESR1 (0.45) ESR1ESR2ARVDR
SCHEMBL3393109 0.69 ESR1 (0.53) ESR1ESR2ARVDRHDAC3
SCHEMBL3392743 0.68 ESR1 (0.45) ESR1ESR2ARVDRHDAC3
SCHEMBL15076980 0.67 ESR1 (0.47) ESR1ESR2ARVDRHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601850-B2 less hypercalcemic than 1a,25 dihydroxy vitamin D3; bone disorders, psoriasis ELI LILLY AND COMPANY (US) 2009-10-13 US disclosed