SCHEMBL13679388

SCHEMBL13679388

Cc1nc(Cl)c(Cl)n1Cc1sc2c(c1C(=O)NCCCO)c(=O)n(C)c(=O)n2C(C)C

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SLC16A1 P53985 7/20 0.53
CYP2C9 P11712 6/20 0.53
CYP3A4 P08684 3/20 0.53
ABCB11 O95342 1/20 0.53
KCNH2 Q12809 1/20 0.30
HTR4 Q13639 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3829699 0.85 SLC16A1 (0.59) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL4803812 0.84 SLC16A1 (0.61) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL4802452 0.80 SLC16A1 (0.80) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL14139859 0.78 SLC16A1 (0.57) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL14099967 0.76 SLC16A1 (0.59) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL4801966 0.75 SLC16A1 (0.75) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL3829224 0.73 SLC16A1 (0.76) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL5791248 0.73 SLC16A1 (0.63) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL3829809 0.73 SLC16A1 (0.78) SLC16A1CYP2C9CYP3A4ABCB11
SCHEMBL3827135 0.72 SLC16A1 (0.61) SLC16A1CYP2C9CYP3A4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414825-B9 THIENOPYRIMIDINEDIONES AND THEIR USE IN THE MODULATION OF AUTOIMMUNE DISEASE ASTRAZENECA AB (SE) 2009-09-16 EP disclosed