SCHEMBL13679405

SCHEMBL13679405

CCn1c(=O)c2c(C(=O)N3C[C@H](O)CO3)c(-c3c(C)n[nH]c3C)sc2n(C(C)C)c1=O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.54
CYP2C9 P11712 5/20 0.54
SLC16A1 P53985 5/20 0.54
SLC16A3 O15427 1/20 0.54
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3826419 0.87 SLC16A1 (0.72) CYP3A4CYP2C9SLC16A1SLC16A3ADORA2B
SCHEMBL3827907 0.78 SLC16A1 (0.80) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3827911 0.78 SLC16A1 (0.80) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL4840916 0.72 SLC16A1 (0.51) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL23958362 0.70 SLC16A1 (1.00) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3826454 0.70 SLC16A1 (1.00) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3826451 0.70 SLC16A1 (1.00) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3828105 0.70 SLC16A1 (0.82) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3828110 0.70 SLC16A1 (0.82) CYP3A4CYP2C9SLC16A1SLC16A3
SCHEMBL3827786 0.70 SLC16A1 (0.74) CYP3A4CYP2C9SLC16A1SLC16A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414825-B9 THIENOPYRIMIDINEDIONES AND THEIR USE IN THE MODULATION OF AUTOIMMUNE DISEASE ASTRAZENECA AB (SE) 2009-09-16 EP disclosed