SCHEMBL13680490

SCHEMBL13680490

Cc1ccc(-c2ccc(NC(=O)OC(C)(C)C)cc2)o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 1/20 0.54
CA12 O43570 1/20 0.51
CA1 P00915 1/20 0.51
CA9 Q16790 1/20 0.51
PRKDC P78527 1/20 0.51
CYP17A1 P05093 3/20 0.50
MEN1 O00255 2/20 0.48
ALDH1A1 P00352 2/20 0.48
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48
RAB9A P51151 1/20 0.48
HDAC1 Q13547 6/20 0.47
HDAC3 O15379 4/20 0.47
HDAC2 Q92769 3/20 0.47
HDAC8 Q9BY41 3/20 0.47
HDAC6 Q9UBN7 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680486 0.85 MAPT (0.52) MEN1ALDH1A1MAPTKMT2AKDM4E
SCHEMBL30175854 0.83 CYP17A1 (0.54) PSMB8CA12CA1CA9PRKDC
SCHEMBL4903830 0.83 CYP17A1 (0.54) PSMB8CA12CA1CA9PRKDC
SCHEMBL2030467 0.83 CYP17A1 (0.54) PSMB8CA12CA1CA9PRKDC
SCHEMBL29957607 0.82 PSMB8 (0.51) PSMB8CA12CA1CA9PRKDC
SCHEMBL14923530 0.82 CA12 (0.46) PSMB8CA12CA1CA9PRKDC
SCHEMBL20865536 0.81 CYP17A1 (0.68) PSMB8CA12CA1CA9PRKDC
SCHEMBL6816610 0.80 KLK7 (0.71) PSMB8CA12CA1CA9CYP17A1
SCHEMBL13680609 0.80 HDAC1 (0.47) CA1ALDH1A1KDM4EGAAHPGD
SCHEMBL13055402 0.79 CYP17A1 (0.59) PSMB8CA12CA1CA9CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed