SCHEMBL13680680

SCHEMBL13680680

Cc1cccc(-c2cnc(-c3ccccc3)nc2)n1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.54
RAB9A P51151 3/20 0.53
NPC1 O15118 2/20 0.53
NFKB1 P19838 2/20 0.53
NFKB2 Q00653 2/20 0.53
RELA Q04206 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
CCR1 P32246 1/20 0.52
CCR8 P51685 1/20 0.52
TGFBR1 P36897 1/20 0.50
HPGDS O60760 7/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.42
METAP2 P50579 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29963679 0.82 MEN1 (0.68) CYP2A6RAB9ANPC1NFKB1SMN1; SMN2
SCHEMBL647992 0.82 MEN1 (0.68) CYP2A6RAB9ANPC1NFKB1SMN1; SMN2
SCHEMBL16189026 0.81 MEN1 (0.56) CYP2A6RAB9ANPC1CCR1CCR8
SCHEMBL13680679 0.81 CCR1 (0.60) CYP2A6RAB9ACCR1CCR8TGFBR1
Bromide SCHEMBL15901554 0.81 RAB9A (0.65) CYP2A6RAB9ANPC1NFKB1SMN1; SMN2
SCHEMBL12594495 0.80 MEN1 (0.64) CYP2A6RAB9ANPC1CCR1CCR8
SCHEMBL17932287 0.80 MEN1 (0.54) CYP2A6RAB9ANPC1CCR1CCR8
SCHEMBL16189330 0.80 MEN1 (0.54) CYP2A6RAB9ANPC1CCR1CCR8
SCHEMBL16189443 0.80 MEN1 (0.54) CYP2A6RAB9ANPC1CCR1CCR8
SCHEMBL19009574 0.80 MEN1 (0.47) CYP2A6RAB9ANPC1NFKB1NFKB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed