SCHEMBL13680744

SCHEMBL13680744

Cc1csc(-c2cnc(C)nc2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.53
CYP2E1 P05181 1/20 0.53
CYP2A6 P11509 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2B6 P20813 1/20 0.53
PDE10A Q9Y233 1/20 0.46
NOS1 P29475 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AOC3 Q16853 2/20 0.38
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HPGDS O60760 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680738 0.84 CYP3A4 (0.50) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680739 0.82 ADORA2A (0.49) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680740 0.81 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680746 0.81 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13680615 0.81 CYP2E1 (0.47) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL15858765 0.81 CYP3A4 (0.47) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL6840352 0.80 CYP3A4 (0.64) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13662750 0.80 CDC25A (0.39) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13681267 0.80 CYP3A4 (0.46) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6
SCHEMBL13681317 0.80 CYP3A4 (0.46) CYP3A4CYP2E1CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed