SCHEMBL13684331

SCHEMBL13684331

COC(=O)C[CH]C1CCC(C(C)(C)C)CC1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.38
APOBEC3A P31941 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
LIPA P38571 1/20 0.36
CYP19A1 P11511 1/20 0.35
MAPT P10636 2/20 0.35
GAA P10253 1/20 0.35
EPHX2 P34913 3/20 0.33
ALDH1A1 P00352 2/20 0.33
GLA P06280 1/20 0.33
HSD11B1 P28845 1/20 0.33
OPRL1 P41146 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7777844 0.73 LIPA (0.54) EPHX1APOBEC3AAPOBEC3GHTTKDM4E
SCHEMBL11058892 0.71 EPHX2 (0.39) EPHX1MAPTEPHX2
SCHEMBL13008729 0.69 LIPA (0.50) EPHX1APOBEC3AAPOBEC3GHTTKDM4E
SCHEMBL11960583 0.67 OPRL1 (0.42) EPHX1APOBEC3AAPOBEC3GHTTSMN1; SMN2
SCHEMBL18334865 0.67 CYP19A1 (0.42) EPHX1APOBEC3AAPOBEC3GHTTKDM4E
SCHEMBL14436583 0.66 SMN1; SMN2 (0.49) EPHX1KDM4ESMN1; SMN2MAPTGAA
SCHEMBL10267770 0.66 SMN1; SMN2 (0.49) EPHX1KDM4ESMN1; SMN2MAPTGAA
SCHEMBL7112401 0.66 TSHR (0.39) EPHX1APOBEC3AAPOBEC3GHTTKDM4E
SCHEMBL2657093 0.66 SMN1; SMN2 (0.49) EPHX1KDM4ESMN1; SMN2MAPTGAA
SCHEMBL24425896 0.66 CYP4F2 (0.35) SMN1; SMN2GAAEPHX2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2522669-A1 3-Spirocyclic indolyl derivatives useful as ORL-1 receptor modulators Janssen Pharmaceutica NV (BE) 2012-11-14 EP disclosed