Formic Acid

Formic Acid

SCHEMBL13685474

COc1ccc(C2(c3ccc(F)c(-c4cccnc4Cl)c3)COC(N)=N2)cc1Cl.O=CO

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.48
CTSD P07339 16/20 0.48
BACE2 Q9Y5Z0 3/20 0.40
REN P00797 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL13685475 1.00 BACE1 (0.48) BACE1CTSDBACE2REN
Formic Acid SCHEMBL2286944 0.87 BACE1 (0.56) BACE1CTSD
Formic Acid SCHEMBL2286466 0.87 BACE1 (0.54) BACE1CTSDBACE2
Formic Acid SCHEMBL2284430 0.85 BACE1 (0.63) BACE1CTSD
Formic Acid SCHEMBL2285584 0.84 BACE1 (0.58) BACE1CTSDBACE2REN
Formic Acid SCHEMBL2285183 0.82 BACE1 (0.53) BACE1CTSDBACE2REN
SCHEMBL2281795 0.82 BACE1 (0.58) BACE1CTSDBACE2
SCHEMBL2281803 0.82 BACE1 (0.58) BACE1CTSDBACE2
SCHEMBL2284420 0.81 BACE1 (0.61) BACE1CTSD
SCHEMBL2284415 0.81 BACE1 (0.61) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2245019-B1 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-11-14 EP disclosed