SCHEMBL13686153

SCHEMBL13686153

COC(=O)CNC(=O)C(C)=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TET2 Q6N021 1/20 0.67
RECQL P46063 1/20 0.52
GAA P10253 2/20 0.46
MGAM O43451 1/20 0.46
SI P14410 1/20 0.46
MGAM2 Q2M2H8 1/20 0.46
TSHR P16473 5/20 0.43
EGLN1 Q9GZT9 1/20 0.43
HSD17B10 Q99714 3/20 0.42
KDM4E B2RXH2 2/20 0.41
EPHX2 P34913 1/20 0.41
ALOX5 P09917 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CA12 O43570 2/20 0.36
CA2 P00918 2/20 0.36
CA14 Q9ULX7 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2523171 0.84 TET2 (0.59) TET2RECQLGAAMGAMSI
SCHEMBL2523319 0.84 TET2 (0.59) TET2RECQLGAAMGAMSI
SCHEMBL2523170 0.84 TET2 (0.59) TET2RECQLGAAMGAMSI
SCHEMBL17589193 0.81 TET2 (0.61) TET2RECQLGAAMGAMSI
SCHEMBL18039446 0.80 TET2 (0.67) TET2RECQLGAAMGAMSI
SCHEMBL3700532 0.80 TET2 (1.00) TET2RECQLGAAMGAMSI
SCHEMBL24112258 0.79 GAA (0.55) TET2GAAMGAMSIMGAM2
SCHEMBL468803 0.79
SCHEMBL26364107 0.79 TET2 (0.53) TET2RECQLGAAMGAMSI
SCHEMBL13962611 0.78 TET2 (0.52) TET2RECQLGAAMGAMSI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592419-B2 Macrocyclic inhibitors of hepatitis C virus NS3-serine protease SCHERING CORPORATION (US) 2009-09-22 US disclosed