SCHEMBL13690840

SCHEMBL13690840

Nc1ccc(N2C3CCC2CC(N)C3)nc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.40
PTPN11 Q06124 16/20 0.39
MAPK3 P27361 1/20 0.39
MAPK1 P28482 1/20 0.39
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12861202 0.78 KDM4E (0.48) RET
SCHEMBL1021345 0.78 RET (0.47) RETPTPN11
SCHEMBL2424922 0.77 HSP90AA1 (0.53) HSP90AA1HSP90AB1
SCHEMBL2424920 0.77 HSP90AA1 (0.53) HSP90AA1HSP90AB1
SCHEMBL31726067 0.77 GRIN2D (0.38) PTPN11GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL2425371 0.76 HSP90AA1 (0.51) RETHSP90AA1HSP90AB1
SCHEMBL3975551 0.76 HSP90AA1 (0.39) RETPTPN11MAPK3MAPK1HSP90AA1
SCHEMBL2424112 0.76 HSP90AA1 (0.52) RETHSP90AA1HSP90AB1
SCHEMBL2612628 0.76 GPR119 (0.41) RET
SCHEMBL1021398 0.76 MAPT (0.52) MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009114173-A1 AZABICYCLO [3. 2. I] OCTYL DERIVATIVES AS 11 BETA-HSDL MODULATORS EXELIXIS, INC. (US) 2009-09-17 WO disclosed