SCHEMBL13699785

SCHEMBL13699785

Bc1cc(Br)cc2c1c(C(=O)NCC13CCC(CC1)CC3)cn2C

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.34
CNR2 P34972 4/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
MAP2K1 Q02750 1/20 0.32
IL1B P01584 1/20 0.31
CNR1 P21554 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1020287 0.89 P2RX7 (0.37) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL1021114 0.88 P2RX7 (0.37) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL13672991 0.88 CNR2 (0.35) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL1019586 0.88 MAP2K1 (0.39) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL1020087 0.88 P2RX7 (0.41) P2RX7IL1B
SCHEMBL13672993 0.82 P2RX7 (0.39) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL13672957 0.81 CNR2 (0.35) P2RX7CNR2MEN1ALDH1A1KMT2A
SCHEMBL13673001 0.81 P2RX7 (0.43) P2RX7IL1B
SCHEMBL1022004 0.81 P2RX7 (0.39) P2RX7IL1B
SCHEMBL1020253 0.81 P2RX7 (0.36) P2RX7CNR2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2105164-A1 Novel P2X7R antagonists and their use Affectis Pharmaceuticals AG (DE) 2009-09-30 EP disclosed