SCHEMBL13705703

SCHEMBL13705703

N#CC(=O)c1cc2[nH]c(=O)c3cnc(C4CCCCC4)n3c2cc1Cl

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 9/20 0.73
PDE5A O76074 3/20 0.64
GRIA1 P42261 2/20 0.33
GRIA2 P42262 2/20 0.33
GRIA3 P42263 2/20 0.33
GRIA4 P48058 2/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
AURKA O14965 1/20 0.32
JAK2 O60674 1/20 0.32
JAK1 P23458 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3579453 0.88 PDE9A (0.78) PDE9APDE5AGRIA1GRIA2GRIA3
SCHEMBL3599970 0.84 PDE9A (0.80) PDE9APDE5AMEN1POLBKMT2A
SCHEMBL3492217 0.84 PDE9A (1.00) PDE9APDE5AGRIA1GRIA2GRIA3
SCHEMBL3592989 0.84 PDE9A (0.80) PDE9APDE5AMEN1POLBKMT2A
SCHEMBL3591571 0.84 PDE9A (0.72) PDE9APDE5AGRIA1GRIA2GRIA3
SCHEMBL3599726 0.82 PDE9A (0.84) PDE9APDE5AMEN1POLBKMT2A
SCHEMBL3606047 0.82 PDE9A (0.81) PDE9APDE5AGRIA1GRIA2GRIA3
SCHEMBL3593184 0.82 PDE9A (0.77) PDE9APDE5AAURKAJAK2JAK1
SCHEMBL3591498 0.82 PDE9A (0.72) PDE9APDE5AMEN1POLBKMT2A
SCHEMBL3599103 0.81 PDE9A (0.78) PDE9APDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2103613-A1 QUINOXALINE DERIVATIVE ASKA Pharmaceutical Co., Ltd. (JP) 2009-09-23 EP disclosed