SCHEMBL13711599

SCHEMBL13711599

N#C[C@]1(c2ccc(-c3ccc(N4CC(n5ccnn5)OC4=O)cc3F)cn2)[C@@H]2COC[C@@H]21

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOA P21397 17/20 0.49
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CALML3 P27482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13711511 0.92 MAOA (0.48) MAOACYP3A4CYP2D6CYP2C9CALML3
SCHEMBL13711519 0.92 MAOA (0.47) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL13711514 0.91 MAOA (0.47) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL13711631 0.90 MAOA (0.48) MAOACYP3A4CYP2D6CYP2C9CALML3
SCHEMBL13711512 0.88 MAOA (0.42) MAOACYP3A4CYP2C9CALML3
SCHEMBL13711577 0.87 MAOA (0.45) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL13711576 0.86 MAOA (0.47) MAOACYP3A4CYP2D6CYP2C9CALML3
SCHEMBL13711617 0.86 MAOA (0.44) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL3366625 0.86 MAOA (0.68) MAOACYP3A4CYP2D6CYP2C9
SCHEMBL14012599 0.86 MAOA (0.68) MAOACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582659-B2 Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof MERCK & CO., INC. (US) 2009-09-01 US disclosed