SCHEMBL13714486

SCHEMBL13714486

CC(C)(C)CC(=O)NCc1cnc[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QPCT Q16769 1/20 0.49
QPCTL Q9NXS2 1/20 0.49
CYP2D6 P10635 2/20 0.47
HRH4 Q9H3N8 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
HPGD P15428 1/20 0.45
CYP3A4 P08684 2/20 0.45
TSHR P16473 2/20 0.45
ALDH1A1 P00352 2/20 0.45
GABRA1 P14867 1/20 0.45
NFKB1 P19838 1/20 0.45
GABRR1 P24046 1/20 0.45
GABRR2 P28476 1/20 0.45
GABRA5 P31644 1/20 0.45
GABRB2 P47870 1/20 0.45
GABRA4 P48169 1/20 0.45
CYP2C19 P33261 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
PMP22 Q01453 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19413331 0.81 QPCT (0.51) QPCTQPCTLCYP2D6HRH4HRH3
SCHEMBL13743314 0.79 CYP3A4 (0.52) QPCTQPCTLCYP2D6HRH4HRH3
SCHEMBL16136337 0.78 QPCT (0.70) QPCTQPCTLCYP2D6HRH4HRH3
SCHEMBL17481129 0.76 QPCT (0.66) QPCTQPCTLCYP2D6HRH4HRH3
SCHEMBL20417155 0.75 QPCT (0.46) QPCTQPCTLHRH4HRH3CYP3A4
SCHEMBL18381403 0.74 TBXAS1 (0.57) QPCTQPCTLCYP2D6HRH4CYP3A4
SCHEMBL19169449 0.72 HPGD (0.57) HPGDCYP3A4ALDH1A1CYP2C19MAPT
SCHEMBL20625835 0.71 HRH3 (0.44) QPCTQPCTLHRH4HRH3
SCHEMBL19413330 0.71 HRH3 (0.44) QPCTQPCTLHRH4HRH3
SCHEMBL13781505 0.69 HPGD (0.66) HPGDALDH1A1KDM4EMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576098-B2 Heterocyclic compounds as inhibitors of factor VIIa BRISTOL-MYERS SQUIBB COMPANY (US) 2009-08-18 US disclosed