SCHEMBL13716079

SCHEMBL13716079

NC(C1CCCCC1)C1CCN(S(=O)(=O)c2cccc3cnccc23)CC1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 12/20 0.77
ROCK1 Q13464 11/20 0.77
PRKD3 O94806 4/20 0.60
PRKCG P05129 4/20 0.60
PRKCB P05771 4/20 0.60
CYP3A4 P08684 4/20 0.60
PRKCA P17252 4/20 0.60
PRKCH P24723 4/20 0.60
PRKCI P41743 4/20 0.60
PRKCE Q02156 4/20 0.60
PRKCQ Q04759 4/20 0.60
PRKCZ Q05513 4/20 0.60
PRKCD Q05655 4/20 0.60
PRKD1 Q15139 4/20 0.60
PRKACA P17612 3/20 0.60
PRKACG P22612 3/20 0.60
PRKACB P22694 3/20 0.60
ADORA3 P0DMS8 2/20 0.60
CYP2C19 P33261 2/20 0.60
KDM4E B2RXH2 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20644189 0.87 ROCK2 (1.00) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL17946426 0.87 ROCK2 (1.00) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL190414 0.87 ROCK2 (1.00) ROCK2ROCK1PRKD3PRKCGPRKCB
Hydrochloric Acid SCHEMBL29377359 0.86 ROCK2 (0.98) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL19543804 0.84 ROCK2 (0.83) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL13716157 0.83 ROCK2 (1.00) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL13716058 0.83 ROCK2 (0.78) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL4729640 0.83 ROCK2 (0.74) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL10985139 0.82 ROCK2 (0.77) ROCK2ROCK1PRKD3PRKCGPRKCB
SCHEMBL6916059 0.82 ROCK2 (0.77) ROCK2ROCK1PRKD3PRKCGPRKCB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7572913-B2 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine BIOAXONE THERAPEUTIQUE INC. (CA) 2009-08-11 US disclosed
US-7572913-B2 Inhibitors of Rho kinase; N-Benzyloxycarbonyl-4-[N''-(tert-butyloxycarbonyl)hydrazino]piperidine; 4-{[N''-(tert-butyloxycarbonyl)-N'-(1'-propyl)]hydrazino}piperidine BIOAXONE THERAPEUTIQUE INC. (CA) 2009-08-11 US disclosed