SCHEMBL13727730

SCHEMBL13727730

CCCc1nccc2c(C)cccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.46
CYP2A6 P11509 2/20 0.46
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
NOS2 P35228 1/20 0.40
PSMD14 O00487 1/20 0.40
COPS5 Q92905 1/20 0.40
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
HSP90AB1 P08238 1/20 0.35
KDM4E B2RXH2 3/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14339123 0.80 CYP1A2 (0.48) CYP1A2CYP2A6HTR1AADRA1DADRA1A
SCHEMBL22113996 0.78 PLAU (0.42) CYP1A2CYP2A6PDE3BPDE3ANOS2
SCHEMBL10245894 0.75 NOS2 (0.45) CYP2A6PDE3BPDE3ANOS2ALDH1A1
SCHEMBL11262866 0.74 PDE3B (0.38) PDE3BPDE3AALDH1A1TSHRKDM4E
SCHEMBL30179063 0.74 CYP2A6 (0.52) CYP2A6PDE3BPDE3ANOS2ALDH1A1
SCHEMBL4066216 0.74 CYP2A6 (0.52) CYP2A6PDE3BPDE3ANOS2ALDH1A1
SCHEMBL11249116 0.73 TDP1 (0.47) CYP1A2PDE3BPDE3AALDH1A1KDM4E
SCHEMBL26538712 0.73 KDM4E (0.48) CYP1A2PDE3BPDE3AHTR1AADRA1D
SCHEMBL8404538 0.72 CYP2A6 (0.59) CYP1A2CYP2A6PDE3BPDE3AHTR1A
SCHEMBL30417914 0.72 CYP1A2 (0.43) CYP1A2CYP2A6HTR1AADRA1DADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603899-B1 HETEROCYCLIC UREA DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2009-08-26 EP disclosed