SCHEMBL13733175

SCHEMBL13733175

CC1(C)CN(C(=O)O)c2cc(C(=O)CC3CC3)cnc21

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
XIAP P98170 14/20 0.37
BIRC2 Q13490 9/20 0.37
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
DRD2 P14416 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
SIGMAR1 Q99720 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27947039 0.85 XIAP (0.34) XIAPBIRC2RXRARXRBRXRG
SCHEMBL13733437 0.82 XIAP (0.36) XIAPBIRC2
SCHEMBL13733640 0.76 XIAP (0.50) XIAPBIRC2
SCHEMBL13732435 0.75 XIAP (0.56) XIAPBIRC2
SCHEMBL13733401 0.73 XIAP (0.36) XIAPBIRC2
Hydrochloric Acid SCHEMBL15649416 0.71 XIAP (0.36) XIAPBIRC2
SCHEMBL13732244 0.69 PDE4D (0.40) XIAPBIRC2
SCHEMBL13732714 0.69 XIAP (0.53) XIAPBIRC2
SCHEMBL13732026 0.68 XIAP (0.64) XIAPBIRC2
SCHEMBL13732143 0.68 XIAP (0.54) XIAPBIRC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699562-A1 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPY Astex Therapeutics Limited (GB) 2014-02-26 EP disclosed
WO-2012143726-A1 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPY ASTEX THERAPEUTICS LIMITED (GB) 2012-10-26 WO disclosed