SCHEMBL13733640

SCHEMBL13733640

CC1(C)CN(C(=O)O)c2cc(C(=O)c3ccccc3)cnc21

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
XIAP P98170 9/20 0.50
BIRC2 Q13490 6/20 0.50
VNN1 O95497 4/20 0.39
PIK3CA P42336 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
NOTUM Q6P988 1/20 0.38
ALDH1A1 P00352 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALOX5 P09917 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22810702 0.87 XIAP (0.44) XIAPBIRC2VNN1PIK3CAALOX15
SCHEMBL13733738 0.86 XIAP (0.45) XIAPBIRC2VNN1PIK3CAALOX5
SCHEMBL27929900 0.80 ELANE (0.40) XIAPBIRC2VNN1PIK3CAALOX15
SCHEMBL13733459 0.77 XIAP (0.39) XIAPBIRC2
SCHEMBL13736703 0.76 XIAP (0.54) XIAPBIRC2
SCHEMBL13735158 0.75 XIAP (0.58) XIAPBIRC2NOTUM
SCHEMBL31725766 0.73 NOTUM (0.44) NOTUMALDH1A1TDP1
SCHEMBL13731600 0.72 KMT2A (0.40) XIAPBIRC2VNN1ALOX15HTT
SCHEMBL22798072 0.68 XIAP (0.58) XIAPBIRC2NOTUM
SCHEMBL25398418 0.66 NOTUM (0.31) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699562-A1 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPY Astex Therapeutics Limited (GB) 2014-02-26 EP disclosed
WO-2012143726-A1 BICYCLIC HETEROCYCLE COMPOUNDS AND THEIR USES IN THERAPY ASTEX THERAPEUTICS LIMITED (GB) 2012-10-26 WO disclosed