SCHEMBL13747129

SCHEMBL13747129

Cc1nc([C@H]2CC[C@@H](C(F)(F)F)CC2)c(-c2ccc(Cl)cc2)c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.38
ACACB O00763 1/20 0.37
ACACA Q13085 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
PSD A5PKW4 2/20 0.36
PLAT P00750 1/20 0.35
PDE2A O00408 7/20 0.35
TNKS O95271 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
PARP2 Q9UGN5 1/20 0.34
CNR1 P21554 2/20 0.34
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
CNR2 P34972 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13746410 0.89 TYMS (0.39) TYMSACACBACACATRPV1PSD
SCHEMBL13746960 0.87 TYMS (0.39) TYMSACACBACACATRPV1PSD
SCHEMBL13746667 0.87 PDE2A (0.37) TYMSPDE2A
SCHEMBL4192359 0.87 PSD (0.38) TYMSACACBACACATRPV1PSD
SCHEMBL13746092 0.87 PSD (0.38) TYMSACACBACACATRPV1PSD
SCHEMBL13746941 0.85 EIF4E (0.36) TYMSACACBACACAPSDPLAT
SCHEMBL13746898 0.85 HSD11B1 (0.39) PSDPDE2A
SCHEMBL13747128 0.85 PLAT (0.34) ACACBACACAPSDPLATPDE2A
SCHEMBL4023129 0.85 PDE2A (0.37) TYMSPDE2A
SCHEMBL4023133 0.85 PDE2A (0.37) TYMSPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed