SCHEMBL13748846

SCHEMBL13748846

CC(C)c1ccc2c(CN(C)CCCN3CCC(C4=CCCS4)(N(C)C)CC3)c[nH]c2c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 11/20 0.38
HTR1B P28222 11/20 0.38
OPRM1 P35372 1/20 0.34
OPRL1 P41146 1/20 0.34
BCHE P06276 4/20 0.33
ACHE P22303 4/20 0.33
TACR2 P21452 2/20 0.32
SIGMAR1 Q99720 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3427309 0.83 OPRM1 (0.42) HTR1DHTR1BOPRM1OPRL1BCHE
SCHEMBL3408690 0.79 OPRL1 (0.49) HTR1DHTR1BOPRM1OPRL1BCHE
SCHEMBL3431374 0.67 HTR1D (0.39) HTR1DHTR1BOPRM1OPRL1
SCHEMBL20883581 0.66 HTR1D (0.57) HTR1DHTR1B
SCHEMBL27816680 0.66 HTR1D (0.67) HTR1DHTR1B
SCHEMBL3431375 0.66 OPRM1 (0.40) HTR1DHTR1BOPRM1OPRL1
SCHEMBL3410692 0.65 OPRL1 (0.65) OPRM1OPRL1BCHEACHESIGMAR1
SCHEMBL27816746 0.62 HTR1D (0.65) HTR1DHTR1BTACR2
SCHEMBL23612450 0.61 HTR1D (0.51) HTR1DHTR1B
SCHEMBL13748790 0.61 HSD17B10 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009103552-A1 SUBSTITUTED INDOLE DERIVATIVES Grünenthal GmbH (DE) 2009-08-27 WO disclosed