SCHEMBL13754649

SCHEMBL13754649

C[C@H](Cc1cccc(CC(=O)NCCc2ccccc2)c1)NC[C@H](CC(C)(C)[Si](C)(C)O)c1ccc(O)c(CO)c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 19/20 0.61
CHRM3 P20309 2/20 0.43
ADRA1D P25100 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
HSD17B2 P37059 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13754578 0.95 ADRB2 (0.54) ADRB2CHRM3
SCHEMBL13754674 0.95 ADRB2 (0.53) ADRB2CHRM3ADRA1DCA1CA2
SCHEMBL13754626 0.94 ADRB2 (0.55) ADRB2CHRM3CA1CA2HSD17B2
SCHEMBL13754576 0.93 ADRB2 (0.71) ADRB2CHRM3
SCHEMBL13754573 0.91 ADRB2 (0.61) ADRB2CHRM3
SCHEMBL13754553 0.90 ADRB2 (0.51) ADRB2CHRM3CA1CA2
SCHEMBL13754624 0.90 ADRB2 (0.64) ADRB2
SCHEMBL14429837 0.90 ADRB2 (0.52) ADRB2CHRM3
SCHEMBL14429835 0.89 ADRB2 (0.58) ADRB2CHRM3
SCHEMBL13590819 0.89 ADRB2 (0.56) ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1624868-B9 \"(2-HYDROXY-2-(4-HYDROXY-3-HYDOXYMETHYLPHENYL)-ETHYLAMINO)- PROPYL]PHENYL DERIVATIVES AS BETA2 AGONISTS PFIZER LTD (GB) 2009-08-12 EP disclosed
US-7268147-B2 Compounds useful for the treatment of diseases PFIZER INC (US) 2007-09-11 US disclosed