SCHEMBL13754663

SCHEMBL13754663

C[C@H](Cc1ccc(CC(=O)OCc2cc(C(F)(F)F)ccc2F)cc1)NC[C@H](O)c1ccc(O)c(CO)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 17/20 0.49
ADRB1 P08588 1/20 0.44
CASP3 P42574 1/20 0.43
CASP6 P55212 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
HIF1A Q16665 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4260356 0.86 ADRB2 (0.62) ADRB2ADRB1
SCHEMBL4255217 0.86 ADRB2 (0.62) ADRB2ADRB1
SCHEMBL14422857 0.81 ADRB2 (0.61) ADRB2ADRB1CASP3CASP6CYP1A2
SCHEMBL4258384 0.80 ADRB2 (0.73) ADRB2ADRB1
SCHEMBL4258388 0.80 ADRB2 (0.73) ADRB2ADRB1
SCHEMBL4388964 0.78 ADRB2 (0.57) ADRB2ADRB1
SCHEMBL4388971 0.78 ADRB2 (0.57) ADRB2ADRB1
SCHEMBL4013045 0.77 ADRB2 (0.69) ADRB2
SCHEMBL4013056 0.77 ADRB2 (0.69) ADRB2
SCHEMBL4255124 0.77 ADRB2 (0.62) ADRB2ADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1624868-B9 \"(2-HYDROXY-2-(4-HYDROXY-3-HYDOXYMETHYLPHENYL)-ETHYLAMINO)- PROPYL]PHENYL DERIVATIVES AS BETA2 AGONISTS PFIZER LTD (GB) 2009-08-12 EP disclosed
EP-1624868-B1 \"(2-HYDROXY-2-(4-HYDROXY-3-HYDOXYMETHYLPHENYL)-ETHYLAMINO)- PROPYL]PHENYL DERIVATIVES AS BETA2 AGONISTS PFIZER LTD (GB) 2008-11-12 EP disclosed