SCHEMBL13754875

SCHEMBL13754875

O=C(O)/C(O)=C/c1cc(OCc2ccccc2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
PKM P14618 1/20 0.46
MAOB P27338 3/20 0.46
PTPN1 P18031 1/20 0.45
MAOA P21397 1/20 0.44
NR4A1 P22736 1/20 0.44
NR4A3 Q92570 1/20 0.44
CCNB2 O95067 1/20 0.44
CDK1 P06493 1/20 0.44
CDK4 P11802 1/20 0.44
CCNB1 P14635 1/20 0.44
CCND1 P24385 1/20 0.44
CCNB3 Q8WWL7 1/20 0.44
SMPD1 P17405 1/20 0.44
P4HTM Q9NXG6 1/20 0.43
PLAU P00749 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1564257 1.00 NR4A2 (0.48) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL13754874 0.85 NR1H4 (0.55) NR4A2MEN1KMT2AALDH1A1MAOB
SCHEMBL1564241 0.85 NR1H4 (0.55) NR4A2MEN1KMT2AALDH1A1MAOB
SCHEMBL29992466 0.84 MAOB (0.58) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL19859637 0.84 MAOB (0.58) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL9756901 0.81 ALDH1A1 (0.63) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL9756904 0.81 ALDH1A1 (0.63) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL1562635 0.79 P4HTM (0.58) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL13427738 0.79 P4HTM (0.58) NR4A2MEN1KMT2AKDM4EALDH1A1
SCHEMBL13754943 0.78 NR3C2 (0.50) KDM4EALOX5CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576198-B1 Integrase inhibitors containing aromatic heterocycle derivatives SHIONOGI & CO., LTD. (JP) 2009-08-18 US disclosed
US-7576198-B1 Integrase inhibitors containing aromatic heterocycle derivatives SHIONOGI & CO., LTD. (JP) 2009-08-18 US disclosed