SCHEMBL1375699

SCHEMBL1375699

Fc1cc(F)c(F)c(Nc2n[nH]c3c(F)c(Cl)c(-c4ccccc4)cc23)c1F.Fc1ccc(Nc2n[nH]c3c(F)c(Cl)c(-c4ccccc4)cc23)cc1F

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.52
CDK1 P06493 1/20 0.52
CDK2 P24941 1/20 0.52
TRPA1 O75762 9/20 0.47
GRM4 Q14833 2/20 0.39
ABCG2 Q9UNQ0 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
FADS1 O60427 4/20 0.36
PTGS2 P35354 1/20 0.35
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
KCNQ1 P51787 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2333075 0.94 GSK3B (0.57) GSK3BCDK1CDK2TRPA1GRM4
SCHEMBL2336326 0.92 GSK3B (0.59) GSK3BCDK1CDK2TRPA1FADS1
SCHEMBL1375716 0.85 GSK3B (0.61) GSK3BCDK1CDK2TRPA1FADS1
SCHEMBL6208060 0.84 TRPA1 (0.55) GSK3BCDK1CDK2TRPA1GRM4
SCHEMBL2334773 0.84 GSK3B (0.62) GSK3BCDK1CDK2TRPA1LMNA
SCHEMBL1376062 0.83 GSK3B (0.59) GSK3BCDK1CDK2TRPA1GRM4
SCHEMBL2336289 0.82 GSK3B (0.58) GSK3BCDK1CDK2TRPA1GRM4
SCHEMBL2336016 0.79 GSK3B (0.55) GSK3BCDK1CDK2TRPA1ABCG2
SCHEMBL2332201 0.78 GSK3B (0.57) GSK3BCDK1CDK2ABCG2MAPT
SCHEMBL1378090 0.78 GSK3B (0.53) GSK3BCDK1CDK2TRPA1GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4764168-B2 2011-08-31 JP claimed
EP-1572200-A1 AMINOINDAZOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS Aventis Pharma S.A. (FR) 2005-09-14 EP claimed
WO-2004062662-A1 AMINOINDAZOLE DERIVATIVES AND USE THEREOF AS KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2004-07-29 WO claimed