SCHEMBL1376202

SCHEMBL1376202

Fc1c(Cl)c(-c2ccccc2)cc2c(Nc3ccc(C(F)(F)F)cc3)n[nH]c12.Fc1cc(Nc2n[nH]c3c(F)c(Cl)c(-c4ccccc4)cc23)cc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.49
CDK1 P06493 1/20 0.49
CDK2 P24941 1/20 0.49
GRM4 Q14833 2/20 0.45
TRPA1 O75762 3/20 0.43
ABCG2 Q9UNQ0 3/20 0.41
FADS1 O60427 1/20 0.41
KDR P35968 2/20 0.39
FLT1 P17948 1/20 0.39
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNQ1 P51787 1/20 0.38
SCN5A Q14524 1/20 0.38
DHODH Q02127 4/20 0.38
AURKB Q96GD4 1/20 0.37
EPHX2 P34913 2/20 0.37
EGFR P00533 1/20 0.36
PDGFRB P09619 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2335033 0.96 GSK3B (0.52) GSK3BCDK1CDK2GRM4TRPA1
SCHEMBL2336016 0.93 GSK3B (0.55) GSK3BCDK1CDK2TRPA1ABCG2
SCHEMBL6528861 0.87 CDK1 (0.49) GSK3BCDK1CDK2GRM4TRPA1
SCHEMBL1378090 0.85 GSK3B (0.53) GSK3BCDK1CDK2GRM4TRPA1
SCHEMBL1376062 0.85 GSK3B (0.59) GSK3BCDK1CDK2GRM4TRPA1
SCHEMBL6206393 0.84 TRPA1 (0.51) GSK3BCDK1CDK2GRM4TRPA1
SCHEMBL2334773 0.84 GSK3B (0.62) GSK3BCDK1CDK2TRPA1FADS1
SCHEMBL2338742 0.80 GSK3B (0.57) GSK3BCDK1CDK2EPHX2
SCHEMBL4380398 0.80 GSK3B (0.62) GSK3BCDK1CDK2KDRFLT1
SCHEMBL4485622 0.79 GRM4 (0.53) GSK3BCDK1CDK2GRM4TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4764168-B2 2011-08-31 JP claimed