SCHEMBL13764323

SCHEMBL13764323

CN(C(c1ccc(Cl)c2nc3n(c12)CCCN3c1c(Cl)cc(Cl)cc1Cl)C(F)(F)F)S(=O)(=O)CC(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 18/20 0.48
MAOB P27338 1/20 0.31
ADORA2A P29274 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3759141 0.82 CRHR1 (0.49) CRHR1MAOBADORA2A
SCHEMBL3759062 0.79 CRHR1 (0.51) CRHR1MAOBADORA2A
SCHEMBL3748308 0.79 CRHR1 (0.58) CRHR1MAOBADORA2A
SCHEMBL3730220 0.78 CRHR1 (0.57) CRHR1MAOBADORA2A
SCHEMBL3755214 0.78 CRHR1 (0.57) CRHR1MAOBADORA2A
SCHEMBL3754663 0.76 CRHR1 (0.51) CRHR1MAOBADORA2A
SCHEMBL3746111 0.75 CRHR1 (0.60) CRHR1ADORA2A
SCHEMBL3748326 0.74 CRHR1 (0.61) CRHR1
SCHEMBL13774767 0.74 CRHR1 (0.54) CRHR1MAOBADORA2A
SCHEMBL3759019 0.71 CRHR1 (0.53) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009093747-A1 TRICYCLIC COMPOUNDS HAVING CORTICOTROPIN-RELEASING FACTOR ANTAGONISTIC ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-07-30 WO disclosed