SCHEMBL13765636

SCHEMBL13765636

CCc1c(-c2nc(-c3ccncc3)no2)nnn1-c1ccccc1F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.53
NPC1 O15118 6/20 0.50
RAB9A P51151 5/20 0.50
PKM P14618 1/20 0.50
KMT2A Q03164 1/20 0.50
LMNA P02545 2/20 0.49
MAPT P10636 6/20 0.47
POLB P06746 2/20 0.45
SMN1; SMN2 Q16637 5/20 0.44
ALDH1A1 P00352 2/20 0.44
S1PR1 P21453 1/20 0.44
TTR P02766 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ATM Q13315 1/20 0.42
NFKB1 P19838 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
HSD17B10 Q99714 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
TSHR P16473 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3753002 0.92 MAPT (0.55) TP53NPC1RAB9APKMKMT2A
SCHEMBL10179953 0.89 RAB9A (0.47) TP53NPC1RAB9APKMKMT2A
SCHEMBL10180279 0.87 RAB9A (0.46) TP53NPC1RAB9APKMKMT2A
SCHEMBL3752697 0.86 TP53 (0.70) TP53NPC1RAB9APKMKMT2A
SCHEMBL10181833 0.85 MAPT (0.54) TP53NPC1RAB9APKMKMT2A
SCHEMBL3761084 0.84 NPC1 (0.54) TP53NPC1RAB9APKMKMT2A
SCHEMBL3760855 0.83 NPC1 (0.52) TP53NPC1RAB9APKMKMT2A
SCHEMBL3752826 0.82 MAPT (0.52) TP53NPC1RAB9AMAPTPOLB
SCHEMBL3755950 0.82 MAPT (0.49) TP53NPC1RAB9APKMKMT2A
SCHEMBL10181626 0.81 NPC1 (0.48) TP53NPC1RAB9APKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080663-A1 TRIAZOLE OXADIAZOLES DERIVATIVES MERCK SERONO S.A. (CH) 2009-07-02 WO disclosed