SCHEMBL13765639

SCHEMBL13765639

Cc1ccc(C#N)c(-c2ccnc3[nH]ccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CIT O14578 1/20 0.47
CCNK O75909 5/20 0.47
CDK12 Q9NYV4 5/20 0.47
LRRK2 Q5S007 3/20 0.47
PRKCI P41743 2/20 0.46
NUDT1 P36639 4/20 0.46
JAK2 O60674 2/20 0.46
PRKACA P17612 2/20 0.46
JAK3 P52333 2/20 0.46
PRKCQ Q04759 2/20 0.46
ROCK1 Q13464 2/20 0.46
IGF1R P08069 2/20 0.46
DYRK1B Q9Y463 2/20 0.46
AURKB Q96GD4 2/20 0.46
IKBKB O14920 1/20 0.46
CHUK O15111 1/20 0.46
DAPK3 O43293 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PAK4 O96013 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12127576 0.84 NUDT1 (0.52) CITCCNKCDK12LRRK2PRKCI
SCHEMBL10125124 0.81 AURKB (0.51) CITCCNKCDK12LRRK2PRKCI
SCHEMBL10125110 0.80 LRRK2 (0.58) CITCCNKCDK12LRRK2PRKCI
SCHEMBL12127929 0.80 PRKCI (0.54) CITCCNKCDK12LRRK2PRKCI
SCHEMBL3576055 0.79 CIT (0.53) CITCCNKCDK12LRRK2PRKCI
SCHEMBL2240671 0.75 AURKB (0.71) CITCCNKCDK12LRRK2PRKCI
SCHEMBL78242 0.74 LRRK2 (0.56) CITLRRK2PRKCINUDT1JAK2
SCHEMBL4790144 0.73 IKBKB (0.70) CITCCNKCDK12LRRK2PRKCI
SCHEMBL12127232 0.73 NUDT1 (0.47) CITCCNKCDK12LRRK2PRKCI
SCHEMBL857132 0.72 IKBKB (0.63) CITCCNKCDK12LRRK2PRKCI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009094123-A1 PROTEIN KINASE INHIBITORS AND USE THEREOF MERCK SERONO S.A. (CH) 2009-07-30 WO disclosed